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alpha-Aminoalkylphosphonates as a tool in experimental optimisation of P1 side chain shape of potential inhibitors in S1 pocket of leucine- and neutral aminopeptidases.
- M. Drąg, J. Grembecka, M. Pawełczak, P. Kafarski
- Chemistry, BiologyEuropean journal of medicinal chemistry
- 1 August 2005
Unnatural amino acids increase activity and specificity of synthetic substrates for human and malarial cathepsin C
- M. Poręba, M. Mihelič, M. Drąg
- BiologyAmino Acids
- 1 January 2014
TLDR
Stereoselective synthesis of 1-aminoalkanephosphonic acids with two chiral centers and their activity towards leucine aminopeptidase.
- M. Drąg, M. Pawełczak, P. Kafarski
- ChemistryChirality
- 2003
TLDR
Structure-Guided, Single-Point Modifications in the Phosphinic Dipeptide Structure Yield Highly Potent and Selective Inhibitors of Neutral Aminopeptidases
- S. Vassiliou, Ewelina Węglarz-Tomczak, A. Mucha
- Chemistry, BiologyJournal of medicinal chemistry
- 5 September 2014
TLDR
Individual stereoisomers of phosphinic dipeptide inhibitor of leucine aminopeptidase.
- A. Mucha, M. Lämmerhofer, W. Lindner, M. Pawełczak, P. Kafarski
- ChemistryBioorganic & medicinal chemistry letters
- 1 March 2008
A synthetic method for diversification of the P1' substituent in phosphinic dipeptides as a tool for exploration of the specificity of the S1' binding pockets of leucine aminopeptidases.
- S. Vassiliou, Metaxia Xeilari, A. Mucha
- Chemistry, BiologyBioorganic & medicinal chemistry
- 1 May 2007
A structural insight into the P1S1 binding mode of diaminoethylphosphonic and phosphinic acids, selective inhibitors of alanine aminopeptidases.
- Ewelina Węglarz-Tomczak, Łukasz Berlicki, M. Pawełczak, B. Nocek, A. Joachimiak, A. Mucha
- ChemistryEuropean journal of medicinal chemistry
- 19 July 2016
A phosphonamidate containing aromatic N-terminal amino group as inhibitor of leucine aminopeptidase-design, synthesis and stability.
- A. Mucha, A. Kunert, J. Grembecka, M. Pawełczak, P. Kafarski
- Chemistry, BiologyEuropean journal of medicinal chemistry
- 1 June 2006
The influence of α-aminophosphonic acids on the activity of aminopeptidase from barley seeds—an approach to determine the enzyme specificity
- Bartosz Oszywa, M. Pawełczak, P. Kafarski
- Chemistry, BiologyActa Physiologiae Plantarum
- 12 February 2015
TLDR
Pentapeptides containing two dehydrophenylalanine residues ‐ synthesis, structural studies and evaluation of their activity towards cathepsin C
- R. Latajka, M. Jewgiński, P. Kafarski
- Chemistry, BiologyJournal of peptide science : an official…
- 1 October 2008
TLDR
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