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Thiadiazoles: Progress Report on Biological Activities
The most active thiadiazole derivatives that have shown considerable biological actions such as antimicrobial, anti-inflammatory, anticancer, anticonvulsant, antidepressant, antioxidant, radioprotective and anti-leishmanial are covered.
Synthesis, anticonvulsant and toxicity evaluation of 2-(1H-indol-3-yl)acetyl-N-(substituted phenyl)hydrazine carbothioamides and their related heterocyclic derivatives
Synthesis, anticonvulsant and toxicity evaluation of 2-(1H-indol-3-yl)acetyl-N-(substituted phenyl)hydrazine carbothioamides and their related heterocyclic derivatives A series of new…
Pharmacological and Pharmaceutical Profile of Valsartan: A Review
Valsartan is an orally active Angiotensin II receptor type 1 antagonist which causes reduction in blood pressure and is used in treatment of hypertension.
THIAZOLES: A VALUABLE INSIGHT INTO THE RECENT ADVANCES AND BIOLOGICAL ACTIVITIES
The present review highlights the recently synthesized thiazoles possessing important biological activities.
SEARCH FOR BIOLOGICAL ACTIVE ISATINS: A SHORT REVIEW
This review covers updated information on the most active isatin derivatives that have been reported to show considerable pharmacological actions such as antimicrobial, anticancer, antiviral, anticonvulsant, anti-inflammatory and analgesic.
Synthesis and anticonvulsant properties of 1-(amino-N-arylmethanethio)-3-(1-substituted benzyl-2, 3-dioxoindolin-5-yl) urea derivatives
Analgesic and Antidepressant Activities of Benzothiazole-Benzamides.
- N. Siddiqui, A. Rana, S. A. Khan, W. Ahsan, M. Alam, Sharique Ahmed
- Chemistry, Psychology
- 22 January 2015
Various benzothiazole-benzamides synthesized were evaluated for their analgesic and antidepressant activities. Interestingly, all the compounds showed promising activities against the two screenings.…
Phthalimides: Biological Profile and Recent Advancements
The present review focuses the novel synthesized phthalimides having important biological activities on their antibacterial, antifungal, analgesic, antitumour, anxiolytic and anti HIV-1 activities.
Cytotoxicity and enzymes estimation of some newer benzimidazoles
Compounds 1, 2, 9 and 10 showed minimum cytotoxic concentration (CTC50) at which 50 percent of cancer cell populations were inhibited and are comparable to the standard drug 5- Fluorouracil.
Synthesis of 8-substituted-4-(2/4-substituted phenyl)-2H-[1,3,5]triazino[2,1-b][1,3]benzothiazole-2-thiones and their anticonvulsant, anti-nociceptive, and toxicity evaluation in mice
- N. Siddiqui, A. Rana, Sharique Ahmed
- Chemistry, BiologyJournal of enzyme inhibition and medicinal…
- 16 November 2009
A number of new 8-substituted-4-(2/4-substituted phenyl)-2H-[1,3,5]triazino[2,1-b][1,3]benzothiazole-2-thiones (4a–t) were synthesized and evaluated for their anticonvulsant, anti-nociceptive,…