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- M. Lakshman Naik, Vaishali Humnabadkar, +47 authors Sandeep R Ghorpade
- Journal of medicinal chemistry
- 2014
4-Aminoquinolone piperidine amides (AQs) were identified as a novel scaffold starting from a whole cell screen, with potent cidality on Mycobacterium tuberculosis (Mtb). Evaluation of the minimum… (More)
- Shahul Hameed P, Suresh M Solapure, +46 authors Vasan K. Sambandamurthy
- Nature communications
- 2015
The widespread emergence of Plasmodium falciparum (Pf) strains resistant to frontline agents has fuelled the search for fast-acting agents with novel mechanism of action. Here, we report the… (More)
- Manoj G Kale, Anandkumar Raichurkar, +31 authors Sandeep R Ghorpade
- Journal of medicinal chemistry
- 2013
A pharmacophore-based search led to the identification of thiazolopyridine ureas as a novel scaffold with antitubercular activity acting through inhibition of DNA Gyrase B (GyrB) ATPase. Evaluation… (More)
- Ramesh R Kale, Manoj G Kale, +24 authors Sandeep R Ghorpade
- Bioorganic & medicinal chemistry letters
- 2014
Scaffold hopping from the thiazolopyridine ureas led to thiazolopyridone ureas with potent antitubercular activity acting through inhibition of DNA GyrB ATPase activity. Structural diversity was… (More)
- Shahul Hameed P, Murugan Chinnapattu, +40 authors Sreekanth A Ramachandran
- Journal of medicinal chemistry
- 2014
Whole-cell high-throughput screening of the AstraZeneca compound library against the asexual blood stage of Plasmodium falciparum (Pf) led to the identification of amino imidazoles, a robust starting… (More)
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