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HIV Capsid is a Tractable Target for Small Molecule Therapeutic Intervention
- W. Blair, C. Pickford, S. Butler
- Biology, ChemistryPLoS pathogens
- 1 December 2010
TLDR
Discovery of Ketone-Based Covalent Inhibitors of Coronavirus 3CL Proteases for the Potential Therapeutic Treatment of COVID-19
- R. Hoffman, R. Kania, Barbara Taggart
- Biology, ChemistryJournal of medicinal chemistry
- 22 July 2020
TLDR
Discovery of a Novel Class of Boron-Based Antibacterials with Activity against Gram-Negative Bacteria
- Vincent Hernández, T. Crépin, J. Plattner
- BiologyAntimicrobial Agents and Chemotherapy
- 7 January 2013
TLDR
Boron‐based phosphodiesterase inhibitors show novel binding of boron to PDE4 bimetal center
- Y. Freund, T. Akama, Yasheen Zhou
- Chemistry, BiologyFEBS letters
- 21 September 2012
Synthesis and antimitotic/cytotoxic activity of hemiasterlin analogues.
- J. Nieman, John Coleman, R. Andersen
- Biology, ChemistryJournal of natural products
- 1 February 2003
TLDR
HTI-286, a synthetic analogue of the tripeptide hemiasterlin, is a potent antimicrotubule agent that circumvents P-glycoprotein-mediated resistance in vitro and in vivo.
- F. Loganzo, C. Discafani, L. Greenberger
- Biology, ChemistryCancer research
- 15 April 2003
TLDR
Improved SARS-CoV-2 Mpro inhibitors based on feline antiviral drug GC376: Structural enhancements, increased solubility, and micellar studies
- Wayne Vuong, Conrad Fischer, J. Vederas
- Chemistry, BiologyEuropean Journal of Medicinal Chemistry
- 30 May 2021
Comprehensive in vitro characterization of PD-L1 small molecule inhibitors
- A. Ganesan, Marawan Ahmed, K. Barakat
- Biology, ChemistryScientific Reports
- 27 August 2019
TLDR
Bioactivation of Flutamide Metabolites by Human Liver Microsomes
- Ping Kang, D. Dalvie, Evan B. Smith, S. Zhou, A. Deese, J. Nieman
- Biology, ChemistryDrug Metabolism and Disposition
- 1 July 2008
TLDR
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