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Design and synthesis of bioactive adamantane spiro heterocycles.
Heterocyclic rimantadine analogues with antiviral activity.
Novel Lipophilic Acetohydroxamic Acid Derivatives Based on Conformationally Constrained Spiro Carbocyclic 2,6-Diketopiperazine Scaffolds with Potent Trypanocidal Activity
TLDR
Novel acetohydroxamic acid derivatives with potent activity against cultured bloodstream-form Trypanosoma brucei and selectivity indices of >1000 are described and S-Enantiomer 7d was the most active derivative against T. cruzi.
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