F Farouz-Grant

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A series of norbinaltorphimine congeners (2-12) which contain different groups at the N17'-position have been synthesized in order to evaluate the role of N17' in conferring kappa opioid antagonist(More)
The presence of a molecular scaffold to orient a basic group is important for potent and selective kappa opioid antagonist selectivity. An attempt to determine how the geometry of the scaffold(More)
A series of amino acid conjugates (2-6) of naltrindole (1) were synthesized from 7'-carboxynaltrindole (7) in order to obtain delta antagonists that would have minimal access to the central nervous(More)
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