• Publications
  • Influence
Ketopiperazine-based renin inhibitors: optimization of the "C" ring.
A systematic investigation of the S3 sub-pocket activity requirements was conducted. It was observed that linear and sterically small side chain substituents are preferred in the S3 sub-pocket forExpand
  • 33
  • PDF
Evaluation of synthetic coumarins for antiausterity cytotoxicity against pancreatic cancers.
A series of functionalized coumarins were synthesized and evaluated for their capacity to inhibit the resistance to starvation of pancreatic cancer cells. This form of cytotoxicity, termedExpand
  • 13