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- Publications
- Influence
Synthesis and antimicrobial activity of novel 5-(1-adamantyl)-2-aminomethyl-4-substituted-1,2,4-triazoline-3-thiones.
- A. El-Emam, Abdul-Malek S. Al-Tamimi, M. Al-Omar, Khalid A. Alrashood, E. E. Habib
- Chemistry, Medicine
- European journal of medicinal chemistry
- 1 October 2013
The reaction of 5-(1-adamantyl)-4-substituted-1,2,4-triazoline-3-thione 5a,b and 10a,b with formaldehyde solution and various primary aromatic amines or 1-substituted piperazines yielded the… Expand
Synthesis, antimicrobial, and anti-inflammatory activity, of novel S-substituted and N-substituted 5-(1-adamantyl)-1,2,4-triazole-3-thiols
- E. Al-Abdullah, Hanadi H. Asiri, S. Lahsasni, E. E. Habib, T. Ibrahim, A. El-Emam
- Chemistry, Medicine
- Drug design, development and therapy
- 12 May 2014
The reaction of 5-(1-adamantyl)-4-phenyl-1,2,4-triazoline-3-thione (compound 5) with formaldehyde and 1-substituted piperazines yielded the corresponding N-Mannich bases 6a–f. The reaction of… Expand
Synthesis, antimicrobial, and anti-inflammatory activities of novel 2-(1-adamantyl)-5-substituted-1,3,4-oxadiazoles and 2-(1-adamantylamino)-5-substituted-1,3,4-thiadiazoles.
- A. Kadi, N. R. El‐Brollosy, O. Al-Deeb, E. E. Habib, T. Ibrahim, A. El-Emam
- Chemistry, Medicine
- European journal of medicinal chemistry
- 1 February 2007
Reaction of 1-adamantanecarbonyl chloride with certain carboxylic acid hydrazides in pyridine yielded the corresponding N-acyl adamantane-1-carbohydrazide derivatives 3a-j, which were cyclized to the… Expand
Non-classical antifolates. Part 2: synthesis, biological evaluation, and molecular modeling study of some new 2,6-substituted-quinazolin-4-ones.
- Fatmah A. M. Al-Omary, L. Abou-zeid, +7 authors H. El-Subbagh
- Chemistry, Medicine
- Bioorganic & medicinal chemistry
- 15 April 2010
A new series of 2,6-substituted-quinazolin-4-ones was designed, synthesized, and evaluated for their in vitro DHFR inhibition, antimicrobial, and antitumor activities. Compounds 22, 33-37, 39-43, and… Expand
Nonclassical antifolates, part 4. 5-(2-aminothiazol-4-yl)-4-phenyl-4H-1,2,4-triazole-3-thiols as a new class of DHFR inhibitors: synthesis, biological evaluation and molecular modeling study.
- Ghada S Hassan, S. El-Messery, +9 authors H. El-Subbagh
- Chemistry, Medicine
- European journal of medicinal chemistry
- 1 August 2013
A new series of compounds possessing 5-(2-aminothiazol-4-yl)-4-phenyl-4H-1,2,4-triazole-3-thiol skeleton was designed, synthesized, and evaluated for their in vitro DHFR inhibition, antimicrobial,… Expand
Synthesis, antimicrobial and anti-inflammatory activities of novel 5-(1-adamantyl)-1,3,4-thiadiazole derivatives.
- A. Kadi, Ebtehal S. Al-Abdullah, I. A. Shehata, E. E. Habib, T. Ibrahim, A. El-Emam
- Chemistry, Medicine
- European journal of medicinal chemistry
- 1 November 2010
New 1-adamanyl-1,3,4-thiadiazole derivatives namely, 5-(1-adamantyl)-1,3,4-thiadiazoline-2-thione 3, 5-(1-adamantyl)-3-(benzyl- or 4-substituted benzyl)-1,3,4-thiadiazoline-2-thione 4a-d,… Expand
Biotechnological applications of quorum sensing inhibition as novel therapeutic strategies for multidrug resistant pathogens.
- M. Shaaban, A. Elgaml, E. E. Habib
- Biology, Medicine
- Microbial pathogenesis
- 1 February 2019
High incidence of antibiotic resistance among bacterial clinical isolates necessitates the discovery of new targets for inhibition of microbial pathogenicity, without stimulation of microbial… Expand
Synthesis, Antimicrobial, and Antiinflammatory Activities of Novel 2‐[3‐(1‐Adamantyl)‐4‐substituted‐5‐thioxo‐1,2,4‐triazolin‐1‐yl]acetic Acids,…
- O. Al-Deeb, M. Al-Omar, N. R. El‐Brollosy, E. E. Habib, T. Ibrahim, A. El-Emam
- Chemistry
- 9 May 2006
Nonclassical antifolates, part 3: synthesis, biological evaluation and molecular modeling study of some new 2-heteroarylthio-quinazolin-4-ones.
- Fatmah A. M. Al-Omary, Ghada S Hassan, S. El-Messery, M. Nagi, E. E. Habib, H. El-Subbagh
- Chemistry, Medicine
- European journal of medicinal chemistry
- 1 May 2013
A new series of 2-heteroarylthio-6-substituted-quinazolin-4-one analogs was designed, synthesized, and evaluated for their in vitro DHFR inhibition, antimicrobial, and antitumor activities. Compounds… Expand
Synthesis, biological evaluation and molecular modeling study of 2-(1,3,4-thiadiazolyl-thio and 4-methyl-thiazolyl-thio)-quinazolin-4-ones as a new class of DHFR inhibitors.
- Sara T. A. Al-Rashood, Ghada S Hassan, +4 authors H. El-Subbagh
- Chemistry, Medicine
- Bioorganic & medicinal chemistry letters
- 15 September 2014
A new series of 2-(1,3,4-thiadiazolyl- or 4-methyl-thiazolyl)thio-6-substituted-quinazolin-4-one analogs was designed, synthesized, and evaluated for their in vitro DHFR inhibition, antimicrobial,… Expand
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