Discovery of thiazolyl-phthalazinone acetamides as potent glucose uptake activators via high-throughput screening.
Synthesis of (±)-Praeruptorin A and Related Khellactone Derivatives
Novel diarylheptanoids as inhibitors of TNF-α production.
Improves Synthesis of (±)-Praeruptorin A and Other Khellactone Esters by Solvent-free DCC Reactions
Esters of 4'-acetylkhellactone such as (+)-praeruptorin A (2) were synthesised in considerably improved yields through use of a low tempeature solvent-free DCC esterification reaction
A novel entry into 1,2,3,4,5,6-hexahydro-3-benzazocine-4,6-dione and 2-substituted-2,5,6,7-tetrahydro-4-benzazonine-1,3-(4H)-dione
Synthesis of 1,4‐disubstituted quinolizidines
Two 9,11-seco-aphylline derivatives and four 4-substitutedimino-1-carbethoxyquinolizidines were synthesized. Conformational assignments of the predominant isomers were derived from spectral data.
ACID-CATALYZED REARRANGEMENT OF 1α,2α-EPOXY-α-TETRAHYDROSANTONIN
SYNTHESIS OF β-EUDESMOL
HL 752: a potent and long-acting antispasmodic agent.