• Publications
  • Influence
Solid phase synthesis of tariquidar-related modulators of ABC transporters preferring breast cancer resistance protein (ABCG2).
Aiming at structural optimization of potent and selective ABCG2 inhibitors, such as UR-ME22-1, from our laboratory, an efficient solid phase synthesis was developed to get convenient access to thisExpand
  • 13
Identification In Silico and In Vitro of Novel Trypanosomicidal Drug‐Like Compounds
Atom‐based bilinear indices and linear discriminant analysis are used to discover novel trypanosomicidal compounds. The obtained linear discriminant analysis‐based quantitative structure–activityExpand
  • 13
  • PDF
Synthesis and Antiparasitic Properties of New 4‐N‐Benzylamino‐4‐Hetarylbut‐1‐enes
New derivatives of 4‐N‐benzylamino‐4‐hetarylbut‐1‐ene containing a pyridyl nucleus were synthesized from benzylamines and pyridine aldehydes. N‐oxide derivatives were obtained from theseExpand
  • 10
A Straightforward Synthetic Approach to Antitumoral Pyridinyl Substituted 7H-Indeno[2,1-c]Quinoline Derivatives Via Three-Component Imino Diels- Alder Reaction
Abstract: A simple and efficient synthetic method of obtaining pyridinyl substituted indeno[2,1- c ]quinolinederivatives has been developed. This method involves a three-component imino Diels-AlderExpand
  • 23
Simulation of spirits distillation for a better understanding of volatile aroma compounds behavior: Application to Armagnac production
Abstract A methodology for the simulation of spirits continuous distillation was developed and applied to the analysis of an Armagnac unit, using the software ProSimPlus®. Distillation data for 66Expand
  • 8
  • PDF
Review and Thermodynamic Modeling with NRTL Model of Vapor-Liquid Equilibria (VLE) of Aroma Compounds Highly Diluted in Ethanol-Water Mixtures at 101.3 kPa
A review of the vapor–liquid equilibrium data of aroma compounds highly diluted in hydroalcoholic mixtures at 101.3 kPa is presented. The study includes 44 aroma compounds present in distilledExpand
  • 5
APLICACION DE LAS REACCIONES DE MULTICOMPONENTES A LA SINTESIS DE INDENO[2,1-c]QUINOLINAS PIRIDIL SUSTITUIDAS Y SINTESIS CONVENCIONAL DE N-(BUTENIL)CLOROALQUILAMIDAS CON FGRAGMENTOS PIRIDINICOS
Las reacciones de multicomponentes, una importante subclase de las reacciones tandem, constan de un proceso ?one-pot? en el cual reaccionan al menos tres componentes que son facilmente asequiblesExpand