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Biocatalysis of the Antimalarial Artemisinin by Mucor ramannianus. Strains
Abstract Biocatalysis of artemisinin by different strains of Mucor ramannianus.* illustrates a simple approach to bioengineering for attaining useful biotransformation strains for preparative orExpand
Hydroxylation of 10-deoxoartemisinin by Cunninghamella elegans.
The microbial metabolism of 10-deoxoartemisinin (1), a derivative of the antimalarial drug artemisinin, was investigated. Various strains of fungi were investigated for their ability to transform 1.Expand
Hydroxylation of 10-deoxoartemisinin to 15-hydroxy-10-deoxoartemisinin by Aspergillus niger
The microbial hydroxylation of 10-deoxoartemisinin was investigated with the aim of obtaining preparative yields of hydroxy derivatives. During 14 d at 28 °C and pH 6.5 Aspergillus niger transformedExpand
Chemoselective reductive alkylation of ammonia with carbonyl compounds: synthesis of primary and symmetrical secondary amines
An efficient, general procedure for highly chemoselective reductive mono-alkylation of ammonia with ketones is reported. Treatment of ketones with ammonia in ethanol and titanium(IV) isopropoxide,Expand
Fluorous methods for the synthesis of peptides and oligonucleotides.
  • B. Miriyala
  • Chemistry, Medicine
  • Topics in current chemistry
  • 2012
The non-covalent affinity of a perfluoro chain towards similar has been exploited by many to separate fluorous tagged compounds from non-fluorous compounds by F-SPE or F-LLE. This purificationExpand
An Efficient and Rapid Synthesis of β-Carboxamide Derivatives using 2,2-dimethyl-2H,4H-1,3-dioxin-4-ones by Microwave Irradiation
Abstract A general, efficient and rapid method for the synthesis of various β-carboxamide derivatives using microwave irradiation is described. Excellent isolated yields were obtained in very shortExpand
Interactions of an Antimicrobial Peptide (Ac-RRWWRF-NH2) and Surfactants: Towards Antimicrobial Peptide Additives for Coatings Applications
Abstract Waterborne coatings are complex formulations containing a number of components to aid stabilization and eventual coalescence of the polymer particles. Almost all systems contain a number ofExpand
Fluorous synthesis of substituted sclerotigenin library.
A fluorous linker-assisted synthetic protocol has been developed for preparation of sclerotigenin-type benzodiazepine-quinazolinone library containing 144 analogues. Amide coupling of fluorousExpand