Share This Author
Synthetic applications of o- and p-halobenzyl sulfones as zwitterionic synthons: preparation of ortho-substituted cinnamates and biarylacetic acids.
Two sequential functionalization processes are applied to the synthesis of ortho-substituted cinnamates and pharmaceuticals belonging to the family of p-biarylacetic acids such as 4-biphenylacetic acid, namoxyrate, xenyhexenic acid, and biphenylpropionic acid.
Lithiated β-aminoalkyl sulfones as mono and dinucleophiles in the preparation of nitrogen heterocycles: Application to the synthesis of capsazepine
N-Boc-α-tosylsarcosine ethyl ester: An α-amido sulfone for the regio- and stereoselective synthesis of protected γ,δ-unsaturated N-methyl-α-amino acids by palladium-catalyzed nucleophilic substitution
P2-Et-Mediated Deprotonation of ortho-Halobenzyl Sulfones: Synthetic Applications as Zwitterionic Synthons
Convergent asymmetric synthesis of indolizidines from (S)-5-(tosylmethyl)-2-pyrrolidinone: synthesis of (−)-δ-coniceine
P2‐Et‐Mediated Deprotonation of ortho‐Halobenzyl Sulfones: Synthetic Applications as Zwitterionic Synthons.
1,3-Dipolar Cycloaddition Reactions with Azomethine Ylides Catalysed by Ag(I). Synthesis of Substituted Prolines
The study of the stereochemistry of substituted prolines, synthesised by 1,3-dipolar cycloaddition reactions between azomethine ylides and alkenes employing substoichiometric amounts of Ag(I) is…
Lithiated β‐Aminoalkyl Sulfones as Mono and Dinucleophiles in the Preparation of Nitrogen Heterocycles: Application to the Synthesis of Capsazepine.
Convergent Asymmetric Synthesis of Indolizidines from (S)‐5‐(Tosylmethyl)‐2‐pyrrolidinone: Synthesis of (‐)‐δ‐Coniceine.