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[125I]RTI-55: a potent ligand for dopamine transporters.
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New, potent cocaine analogs: ligand binding and transport studies in rat striatum.
Two potent cocaine analogs have been developed that have the highest known affinities for the cocaine binding site in rat striatum. Both 3 beta-(4-chlorophenyl)- (RTI-COC-31) and 3Expand
  • 67
Peptide derivatives of primaquine as potential antimalarial agents.
Three peptide derivatives of primaquine were synthesized. The compounds were tested for radical curative antimalarial activity against Plasmodium cynomolgi in rhesus monkeys and blood schizonticidalExpand
  • 44
Synthesis of some 17-substituted 3,10-ethano-5alpha-estranes.
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Isothiocyanate derivatives of cocaine: irreversible inhibition of ligand binding at the dopamine transporter.
Isothiocyanate derivatives of (-)-cocaine were prepared and tested for inhibitory potency at the cocaine receptor in rat striatal membranes. Coincubation with m-isothiocyanatobenzoylecgonine methylExpand
  • 34
High Potency Cocaine Analogs: Neurochemical, Imaging, and Behavioral Studies
Recent evidence suggests the behavioral properties of cocaine are related to its ability to inhibit dopamine (DA) reuptake.1.2 Specific binding sites tbr cocaine have been identified with a host ofExpand
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Reduced 8-aminoquinoline analogues as potential antimalarial agents.
The synthesis of 1-alkyl-8-(aminoalkylamino)-6-methyl1-1,2,3,4-tetrahydroquinolines, 8-(4'-amino-1'-methylbutylamino)-6-methoxy-1-methyl1-1,2-dihydroquinoline, 5-substitutedExpand
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